I-Modafinil (i-Provigil) isetyenziselwa ukuphatha i-apnea yokulala, i-narcolepsy kunye nokunye.
Uninzi lwabantu basebenzise kakubi ukusetyenziswa kwengqondo okanye ukusetyenziswa kweziyobisi zengqondo ezingabonakaliyo ukwenzela ukwandisa umkhiqizo, ukuxhatshazwa kunye nokuncedisa ngemingeni engqondweni. Nangona ukusetyenziswa kakubi kweziyobisi ezinokuphuculwa kwengqondo ezifana ne-amphetamine, i-methylphenidate kunye ne-modafinil (i-Provigil) ngokuqhelekileyo idibene nabafundi baseyunivesiti-ukuqikelelwa kwe-7 ukuya kuma-20 ekhulwini kwabafundi beekholeji zase-US baxelele ukusetyenziswa kakubi kwezidakamizwa - amanye amaqela amangalisayo abantu iziyobisi, nazo.
Ngokomzekelo, ama-8.9 eepesenti zabagqirha abaphandwayo eJamani babika ukusetyenziswa okungagqirwanga kokusetyenziswa kweziyobisi eziphuculisayo.
I-Modafinil imele ukuba ibe ngumlutha ongaphantsi kunezinye i-psychostimulants ezifana ne-amphetamine; Nangona kunjalo, asiyiqondi kakuhle ukuba le nkunkuma isebenza njani okanye igalelo layo elide. Ukongezelela, i-modafinil inokubangela ukuba kube nemiphumo embi kakhulu kwaye kufuneka ithathwe kuphela xa imiselwe ngugqirha.
Yintoni i Modafinil?
Ngezinye izikhathi i-Modafinil ibizwa ngokuba yi-"agent-promoting agent". Abaphandi bakholelwa ukuba le nkunkuma isebenza ngokwandisa ukutholakala kwe-synaptic ye-neurotransmitters njenge-monoamines, i-catecholamines, i-dopamine, i-serotonin, i-adenosine, i-histamine kunye ne-noradrenaline. I-Modafinil ithinta i-hypothalamus, i-hippocampus, kunye ne-amygdala eziyinxalenye yengqondo.
I-Modafinil yipilisi esetyenziswe ngomlomo ngokuphindaphindiweyo ngemini. Uninzi lwabantu abasebenza emini bathatha isigqirha kusasa malunga nesisu esipheleleyo okanye esingenalutho.Nokho, abasebenzi abashintshayo ukuba bathathe isilwanyana ukuze baphakamise ukuvuka baphathe izidakamizwa ngaphambi kokuba iinguqu zabo ziqale.
Yenzani i-Modafinil?
I-Modafinil isetyenziselwa ukuphatha iingxaki ngokuqonda, ukuvusa, nokuvuka. Ezinye iimeko eziphathwe nge-modafinil ziquka ezi zilandelayo:
- Ukunqongophala
- Isifo sokulala seShift-work
- Ukukhubazeka kokulala kokugula
- Ukulimala kwengqondo ebuhlungu
- Ulwaphulo lwe-Adjuvant of depress
- ADHD
- Unonophelo olusisigxina okanye lokuphela komsebenzi
Ngokubhekiselele ekunakekeleni kwinkqubo yokunyamekela okanye yokuphela komsebenzi, ezininzi iingcali zikhetha ukucacisa iingqondo ezinjenge-modafinil kuba ziphucula iimoya ngokukhawuleza kuneemithi zengqondo. Ukongezelela, ukuxhomekeka kukungakhathazeki ngaphantsi kokunyamekela kokuphela komsebenzi.
Iziphumo ezimbi
Imiphumo emibi kakhulu yeModafinil ibandakanya oku kulandelayo:
- Ukuvutha
- I sizathu
- Ukutshitshiswa
- Ukuxhalabisa
Ezinye iziphumo ezimbi zibandakanya oku kulandelayo:
- Ukungabikho
- Uhudo
- Ukutyunjwa
- Ukuxela
- Ukuthuka
- Ukuphefumula okunzima
- Iintlungu zesifuba
- Intliziyo engavumelekanga
- Iinjongo zokuzibulala (iingcamango zokuzibulala)
- I-hallucination
- Rash
- Blisters
- Iimbuzi
Eminye yale miphumo emibi iyatshitshisa kwaye iyingozi, qiniseka ukuba uqhagamshelane nodokotela wakho ukuba ufumana nawuphi na kubo.
Ukongezelela, ezinye zeziphumo ezinobungozi ezifana nokulala, ukungazinzi, iintlungu zesifuba, isisonguluko, kunye nokudideka kunokubangelwa ukugqithisa ngokwemodafinil. Ukuba ukrokrela ukudlula, fowuni iinkonzo eziphuthumayo okanye uqhagamshelane nodokotela ngokukhawuleza.
Ukungqinelana
I-Modafinil ayilona wonke umntu, kwaye phambi kokuba ugqirha wakho akumisele le nyilisi, umele umxelele oku kulandelayo:
- I-allergies ukuya kwi-modafinil okanye i-armodafinil (i-enantiomer of modafinil)
- Amachiza e-Antidepressant aquka ii-SSRI, ii-TCAs kunye ne- benzodiazepines
- Ukuchithwa kwemithi efana ne-phenytoin ne-carbamazepine
- Amayeza antifungal njenge-itraconazole ne-ketoconazole
- Ukusetyenziswa kakubi kweziyobisi okanye ukuxhomekeka
- IiVithamini, izongezelelo zondlo, kunye nezongezelelo zemfuyo
Abantu abane-angina okanye abasanda kuhlaselwa yintliziyo kufuneka banganikezwa nge-modafinil. Ukongezelela, akucaci ukuba umphumo we-modafinil unesigxina sokuthatha. Ngaloo ndlela, i-modafinil inokuba yingozi kubantu abanesifo sokuhluthwa kunye nokunye ukuphazamiseka kwemithi.
Akukho zifundo zangexesha elide kwimiphumo ye-modafinil ebuchosheni. Ugqirha kufuneka acinge ngenyameko ukuba awanike i-modafinil kwaye ayilinganise inzuzo yeempawu zayo ezikhuthazayo kunye nemiphumo emibi.
Nangona i-modafinil mhlawumbi iyalutha kakhulu kunezinye izikhuthazo ezifana ne-amphetamines kunye ne-methylphenidate, isenokubakhokelela ekuxhomekeke kuyo.
Nceda uqonde ukuba rhoqo xa ugqirha enza isigqibo sokumisela i-modafinil, esi sigqibo sisigulane esithile. Ngamanye amagama, ukuba unikwe i-modafinil okanye enye i-psychostimulant, lo myalelo kuphela kuwe. Akufanele uhlanganyele okanye uthengise i-modafinil-okanye nayiphina imithi yesigqirha kuloo nto. Ukuchithwa okunjalo kuyingozi kwaye akukho mthethweni.
Imithombo
ULu D, uNorman MA, Singh B, uLee K. Uxinzelelo kunye nezinye iingxaki zempilo yengqondo. Ku: Williams BA, Chang A, Ahalt C, Chen H, Conant R, uLandefeld C, Ritchie C, Yukawa M. eds. Ukuxilongwa kwangoku kunye noNyango: i-Geriatrics, udidi lwesiBini . New York, NY: McGraw-Hill; 2014.
Siu G. Pharmacotherapy. Ku: Maitin IB, Cruz E. eds. UKUPHATHWA KWE-CURRENT Ukuxilongwa nokuPhathwa kweMpilo: I-Medicine yePhysical & Rehabilitation . New York, NY: McGraw-Hill; 2015.
Inqaku elibizwa ngokuthi "Ukusetyenziswa kokusetyenziswa kwezinto ezinokwenziwa kwengqondo phakathi kwabafundi base-New Zealand" baseSam Ram kunye nabalobi ababambisene nabo kwi-Drug and Alcohol Review eshicilelwe ngo-2015.